Nϵ-Acryloyllysine Piperazides as Irreversible Inhibitors of Transglutaminase 2 : (Synthesis, Structure-Activity Relationships, and Pharmacokinetic Profiling)

Autor*innen

Wodtke, Robert ; Hauser, Christoph ; Ruiz-Gómez, Gloria ; Jäckel, Elisabeth ; Bauer, David ; Lohse, Martin ; Wong, Alan ; Pufe, Johanna ; Ludwig, Friedrich-Alexander ; Fischer, Steffen ; Hauser, Sandra ; Greif, Dieter ; Pisabarro, M. Teresa ; Pietzsch, Jens ; Pietsch, Markus ; Löser, Reik

DOI

10.1021/acs.jmedchem.8b00286